BDBM50160309 2-[(R)-4-(3-Chloro-pyridin-2-yl)-2-methyl-piperazin-1-yl]-6-methoxy-1H-benzoimidazole::CHEMBL361144

SMILES COc1ccc2nc([nH]c2c1)N1CCN(C[C@H]1C)c1ncccc1Cl

InChI Key InChIKey=QMCSRFHZOUUSFJ-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50160309   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Purdue Pharma

Curated by ChEMBL

LigandBDBM50160309(2-[(R)-4-(3-Chloro-pyridin-2-yl)-2-methyl-piperazi...)Copy SMILESCopy InChI

Affinity DataIC50: 665nMAssay Description:Antagonist activity in capsaicin-induced FLIPR assays in HEK293 cells expressing human TRPV1More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
11/10/2009
Entry Details Article
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