BDBM50160715 CHEMBL3785865

SMILES Cc1c2C(=O)N(Cc3ccccc3-c3ccccc3)C(C(=O)NC(C)(C)C)c2ccc1O

InChI Key InChIKey=FZIZRJKMCCBMMF-UHFFFAOYSA-N

Data  9 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 9 hits for monomerid = 50160715   

LigandPNGBDBM50160715(CHEMBL3785865)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human Kv1.5 channel by Rb-flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2017
Entry Details Article
PubMed
LigandPNGBDBM50160715(CHEMBL3785865)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human Kv1.5 channel by QPatch-clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2017
Entry Details Article
PubMed
LigandPNGBDBM50160715(CHEMBL3785865)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human Kv1.5 channel by QPatch-clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2017
Entry Details Article
PubMed
LigandPNGBDBM50160715(CHEMBL3785865)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human Kv1.5 channel by QPatch-clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2017
Entry Details Article
PubMed
LigandPNGBDBM50160715(CHEMBL3785865)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of human Kv1.5 channel by Rb-flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2017
Entry Details Article
PubMed
LigandPNGBDBM50160715(CHEMBL3785865)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of human Kv1.5 channel by Rb-flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2017
Entry Details Article
PubMed
LigandPNGBDBM50160715(CHEMBL3785865)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2017
Entry Details Article
PubMed
LigandPNGBDBM50160715(CHEMBL3785865)
Affinity DataIC50: 4.60E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2017
Entry Details Article
PubMed
LigandPNGBDBM50160715(CHEMBL3785865)
Affinity DataIC50: 4.60E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2017
Entry Details Article
PubMed