BDBM50171081 CHEMBL3805036

SMILES CN(C)c1ccc2nc(-c3ccccc3)c(cc2c1)-c1ccccc1

InChI Key InChIKey=WZDHUXYPWVWTPR-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50171081   

TargetProteasome subunit beta type-5(Human)
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50171081(CHEMBL3805036)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Michigan State University

Curated by ChEMBL
LigandPNGBDBM50171081(CHEMBL3805036)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of human 20S proteasome chymotryptic-like activity using Suc-LLVY-AMC as substrate assessed as fluorescence quinching control by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed