BDBM50172296 1-Benzenesulfonyl-3-(1,2,5,6-tetrahydro-pyridin-3-yl)-1H-indole::CHEMBL193824

SMILES O=S(=O)(c1ccccc1)n1cc(C2=CCCNC2)c2ccccc12

InChI Key InChIKey=AVLOHBOUEWFHFB-UHFFFAOYSA-N

Data  1 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50172296   

Target5-hydroxytryptamine receptor 6(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50172296(1-Benzenesulfonyl-3-(1,2,5,6-tetrahydro-pyridin-3-...)
Affinity DataKi:  4.60nMAssay Description:Displacement of [3H]LSD from cloned human 5-hydroxytryptamine 6 receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50172296(1-Benzenesulfonyl-3-(1,2,5,6-tetrahydro-pyridin-3-...)
Affinity DataEC50:  159nMAssay Description:Effective concentration for cAMP production in HeLa cells expressing human 5-HT6 receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed