BDBM50172301 1-(4-Fluoro-benzenesulfonyl)-3-(1,2,5,6-tetrahydro-pyridin-3-yl)-1H-indole::CHEMBL194568

SMILES Fc1ccc(cc1)S(=O)(=O)n1cc(C2=CCCNC2)c2ccccc12

InChI Key InChIKey=PKSXYHMBORWHAI-UHFFFAOYSA-N

Data  1 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50172301   

Target5-hydroxytryptamine receptor 6(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50172301(1-(4-Fluoro-benzenesulfonyl)-3-(1,2,5,6-tetrahydro...)
Affinity DataEC50:  345nMAssay Description:Effective concentration for cAMP production in HeLa cells expressing human 5-HT6 receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50172301(1-(4-Fluoro-benzenesulfonyl)-3-(1,2,5,6-tetrahydro...)
Affinity DataKi:  10.5nMAssay Description:Displacement of [3H]LSD from cloned human 5-hydroxytryptamine 6 receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed