BDBM50172313 1-(5-Chloro-thiophene-2-sulfonyl)-3-piperidin-3-yl-1H-indole::CHEMBL371318

SMILES Clc1ccc(s1)S(=O)(=O)n1cc(C2CCCNC2)c2ccccc12

InChI Key InChIKey=JJNCPALKVTYAFB-UHFFFAOYSA-N

Data  1 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50172313   

Target5-hydroxytryptamine receptor 6(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50172313(1-(5-Chloro-thiophene-2-sulfonyl)-3-piperidin-3-yl...)
Affinity DataEC50:  58.5nMAssay Description:Effective concentration for cAMP production in HeLa cells expressing human 5-HT6 receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50172313(1-(5-Chloro-thiophene-2-sulfonyl)-3-piperidin-3-yl...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]LSD from cloned human 5-hydroxytryptamine 6 receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed