BDBM50177117 CHEMBL3814092

SMILES N[C@@H](COP(O)(=O)O[C@@H]1CCCO[C@@H]1COC(=O)CCc1ccccc1OCc1cccc(Oc2ccccc2)c1)C(O)=O

InChI Key InChIKey=BIGHQMOUQYMHQN-UHFFFAOYSA-N

Data  8 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 8 hits for monomerid = 50177117   

TargetPutative P2Y purinoceptor 10(Mouse)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50177117(CHEMBL3814092)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at mouse P2Y10 receptor expressed in HEK293A cells after 1.5 hrs by alkaline phosphatase tagged-TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/15/2017
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 34(Mouse)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50177117(CHEMBL3814092)
Affinity DataEC50:  138nMAssay Description:Agonist activity at mouse GPR34 expressed in HEK293A cells cotransfected with chimeric Galphaq/il after 1.5 hrs by alkaline phosphatase tagged-TGFalp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/15/2017
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 34(Mouse)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50177117(CHEMBL3814092)
Affinity DataEC50:  140nMAssay Description:Agonist activity at mouse GPR34 expressed in HEK293A cells cotransfected with chimeric Galphaq/il after 1.5 hrs by alkaline phosphatase tagged-TGFalp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/15/2017
Entry Details Article
PubMed
TargetPutative P2Y purinoceptor 10(Mouse)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50177117(CHEMBL3814092)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at mouse P2Y10 receptor expressed in HEK293A cells after 1.5 hrs by alkaline phosphatase tagged-TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/15/2017
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 34(Mouse)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50177117(CHEMBL3814092)
Affinity DataEC50:  180nMAssay Description:Agonist activity at mouse GPR34 expressed in HEK293 cells co-transfected with AP-TGFalpha/chimeric Galphaq/i1 assessed as induction of ectodomain she...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 34(Mouse)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50177117(CHEMBL3814092)
Affinity DataEC50:  182nMAssay Description:Agonist activity at mouse GPR34 expressed in HEK293 cells co-transfected with AP-TGFalpha/chimeric Galphaq/i1 assessed as induction of ectodomain she...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 34(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50177117(CHEMBL3814092)
Affinity DataEC50:  150nMAssay Description:Agonist activity at human GPR34 expressed in HEK293 cells co-transfected with AP-TGFalpha/chimeric Galphaq/i1 assessed as induction of AP-TGFalpha re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 34(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50177117(CHEMBL3814092)
Affinity DataEC50:  151nMAssay Description:Agonist activity at human GPR34 expressed in HEK293 cells co-transfected with AP-TGFalpha/chimeric Galphaq/i1 assessed as induction of AP-TGFalpha re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed