BDBM50177163 1-(bis(4-chlorophenyl)methyl)-3-(4-bromophenyl)urea::CHEMBL436309

SMILES Clc1ccc(cc1)C(NC(=O)Nc1ccc(Br)cc1)c1ccc(Cl)cc1

InChI Key InChIKey=OCTCUNGVDUMZHF-UHFFFAOYSA-N

Data  1 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50177163   

TargetCannabinoid receptor 1(Human)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50177163(1-(bis(4-chlorophenyl)methyl)-3-(4-bromophenyl)ure...)
Affinity DataEC50:  700nMAssay Description:Activity at human CB1 receptor by [35S]GTP-gamma-S binding stimulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50177163(1-(bis(4-chlorophenyl)methyl)-3-(4-bromophenyl)ure...)
Affinity DataKi:  1.25E+3nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed