BDBM50177667 CHEMBL3815084

SMILES COC1(COC1)c1nc2c(nc(nc2n1C)-c1cnc(N)nc1)N1CCOCC1

InChI Key InChIKey=LDNVLEUCPIRSSG-UHFFFAOYSA-N

Data  1 KI

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50177667   

TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Genentech

Curated by ChEMBL

LigandBDBM50177667(CHEMBL3815084)Copy SMILESCopy InChI

Affinity DataKi:  5nMAssay Description:Inhibition of recombinant PI3Kalpha (unknown origin) using dioctanoylglycerol-PIP2 as substrate incubated for 30 mins in presence of TAMRA-PIP3 by fl...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
9/16/2017
Entry Details Article
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