BDBM50188027 2-ethoxy-3-(1-(3-(5-methyl-2-phenyloxazol-4-yl)propyl)-1H-indol-4-yl)propanoic acid::CHEMBL213487

SMILES CCOC(Cc1cccc2n(CCCc3nc(oc3C)-c3ccccc3)ccc12)C(O)=O

InChI Key InChIKey=DKDATBYVPQYIRT-UHFFFAOYSA-N

Data  2 IC50  3 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50188027   

TargetPeroxisome proliferator-activated receptor delta(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50188027(2-ethoxy-3-(1-(3-(5-methyl-2-phenyloxazol-4-yl)pro...)
Affinity DataEC50:  2.40E+3nMAssay Description:Activity at PPARdelta by luciferase reporter gene transactivation assay relative to GW 501516More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50188027(2-ethoxy-3-(1-(3-(5-methyl-2-phenyloxazol-4-yl)pro...)
Affinity DataIC50: 274nMAssay Description:Binding affinity to PPARgamma by radio ligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50188027(2-ethoxy-3-(1-(3-(5-methyl-2-phenyloxazol-4-yl)pro...)
Affinity DataIC50: 756nMAssay Description:Binding affinity to PPARalpha by radio ligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50188027(2-ethoxy-3-(1-(3-(5-methyl-2-phenyloxazol-4-yl)pro...)
Affinity DataEC50:  190nMAssay Description:Activity at PPARalpha by luciferase reporter gene transactivation assay relative to farglitazarMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50188027(2-ethoxy-3-(1-(3-(5-methyl-2-phenyloxazol-4-yl)pro...)
Affinity DataEC50:  90nMAssay Description:Activity at PPARgamma by luciferase reporter gene transactivation assay relative to edaglitazoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed