BDBM50188267 (4-methylpiperazin-1-yl)(3-(thiophen-3-yl)-1,4-dihydroindeno[1,2-c]pyrazol-7-yl)methanone::CHEMBL378007

SMILES CN1CCN(CC1)C(=O)c1ccc2Cc3c(n[nH]c3-c3ccsc3)-c2c1

InChI Key InChIKey=XOQLPCMMWXCDHX-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50188267   

TargetVascular endothelial growth factor receptor 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50188267((4-methylpiperazin-1-yl)(3-(thiophen-3-yl)-1,4-dih...)
Affinity DataIC50: 4.08E+6nMAssay Description:Inhibition of VEGF-induced human KDR phosphorylation transfected in NIH3T3 cells by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed