BDBM50194625 (R)-3-{2-methyl-4-[3-(2-phenoxy-4-trifluoromethoxy-phenoxy)-butoxy]-phenyl}-propionic acid::CHEMBL214921

SMILES C[C@H](CCOc1ccc(CCC(O)=O)c(C)c1)Oc1ccc(OC(F)(F)F)cc1Oc1ccccc1

InChI Key InChIKey=CQHWVRVOKKOIJC-UHFFFAOYSA-N

Data  6 IC50  3 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 9 hits for monomerid = 50194625   

LigandPNGBDBM50194625((R)-3-{2-methyl-4-[3-(2-phenoxy-4-trifluoromethoxy...)
Affinity DataEC50:  2nMAssay Description:Transactivation of human PPARdelta in CV1 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194625((R)-3-{2-methyl-4-[3-(2-phenoxy-4-trifluoromethoxy...)
Affinity DataEC50:  5nMAssay Description:Transactivation of human PPARgamma in CV1 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194625((R)-3-{2-methyl-4-[3-(2-phenoxy-4-trifluoromethoxy...)
Affinity DataIC50: 5nMAssay Description:Displacement of [3H]2-(4-{2-[3-(2,4-difluoro-phenyl)-1-heptyl-ureido]-ethyl}-phenoxy)-2-methyl-butyric acid from human PPARdelta by SPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194625((R)-3-{2-methyl-4-[3-(2-phenoxy-4-trifluoromethoxy...)
Affinity DataIC50: 5nMAssay Description:Agonist activity at PPARdeltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
LigandPNGBDBM50194625((R)-3-{2-methyl-4-[3-(2-phenoxy-4-trifluoromethoxy...)
Affinity DataIC50: 6nMAssay Description:Agonist activity at PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
LigandPNGBDBM50194625((R)-3-{2-methyl-4-[3-(2-phenoxy-4-trifluoromethoxy...)
Affinity DataIC50: 6nMAssay Description:Displacement of [3H]2-methyl-2-(4-{3-[propyl-(5-pyridin-2-yl-thiophene-2-sulfonyl)-amino]-propyl}-phenoxy)-propionic acid from human PPARgamma by SPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194625((R)-3-{2-methyl-4-[3-(2-phenoxy-4-trifluoromethoxy...)
Affinity DataEC50:  642nMAssay Description:Transactivation of human PPARalpha in CV1 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194625((R)-3-{2-methyl-4-[3-(2-phenoxy-4-trifluoromethoxy...)
Affinity DataIC50: 897nMAssay Description:Displacement of [3H]2-(4-{2-[3-(2,4-difluoro-phenyl)-1-heptyl-ureido]-ethyl}-phenoxy)-2-methyl-butyric acid from human PPARalpha by SPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194625((R)-3-{2-methyl-4-[3-(2-phenoxy-4-trifluoromethoxy...)
Affinity DataIC50: 897nMAssay Description:Agonist activity at PPARalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed