BDBM50195079 (S)-2-((5-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)pyridin-2-yl)methyl)-tetrahydrofuran-2-carboxylic acid::CHEMBL218487

SMILES Cc1oc(nc1CCOc1ccc(C[C@@]2(CCCO2)C(O)=O)nc1)-c1ccccc1

InChI Key InChIKey=OYWWKKYTRPWVCD-UHFFFAOYSA-N

Data  2 KI  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50195079   

LigandPNGBDBM50195079((S)-2-((5-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)...)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human PPAR alpha in HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195079((S)-2-((5-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)...)
Affinity DataEC50:  26nMAssay Description:Agonist activity at human PPAR gamma in HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195079((S)-2-((5-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)...)
Affinity DataKi:  43nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195079((S)-2-((5-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)...)
Affinity DataKi:  340nMAssay Description:Displacement of radiolabeled GW-2331 from human PPAR alpha by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed