BDBM50197524 CHEMBL3957061

SMILES Cn1ccc(c1)-c1ccc2n(cnc2c1)-c1ccc(CC(=O)Nc2cc(on2)C(C)(C)C)cc1

InChI Key InChIKey=REQJIWOWTBYYLI-UHFFFAOYSA-N

Data  2 Kd

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50197524   

TargetVascular endothelial growth factor receptor 2(Human)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50197524(CHEMBL3957061)
Affinity DataKd: <1nMAssay Description:Binding affinity to of human partial length VGFR2 expressed in mammalian system by active site-directed competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50197524(CHEMBL3957061)
Affinity DataKd: <1nMAssay Description:Binding affinity to of human partial length RET expressed in bacterial system by active site-directed competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2018
Entry Details Article
PubMed