BDBM50198691 CHEMBL3923909

SMILES Fc1ccc(\C=C2/CCCCc3c(nn(c23)-c2ccc(Cl)c(Cl)c2)C(=O)NC2(CC2)c2ccccn2)cc1

InChI Key InChIKey=KLLWBIAQONUJSO-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50198691   

TargetCannabinoid receptor 1(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50198691(CHEMBL3923909)
Affinity DataEC50:  13nMAssay Description:Inverse agonist activity at human cannabinoid receptor 1 expressed in HEK293 cells assessed as increase in forskolin-induced cAMP production preincub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50198691(CHEMBL3923909)
Affinity DataEC50:  807nMAssay Description:Inverse agonist activity at human cannabinoid receptor 2 expressed in HEK293 cells assessed as increase in forskolin-induced cAMP production preincub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed