BDBM50202476 CHEMBL3945688

SMILES COC(=O)COc1ccc2n(Cc3ccccc3C(F)(F)F)c(nc2c1)C(C)c1ccc(CC(C)C)cc1

InChI Key InChIKey=UMPIPJNQFPGAIU-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50202476   

TargetArachidonate 5-lipoxygenase-activating protein(Human)
Gazi University

Curated by ChEMBL
LigandPNGBDBM50202476(CHEMBL3945688)
Affinity DataIC50: 210nMAssay Description:Inhibition of FLAP in human neutrophils assessed as suppression of A23187-stimulated 5-LO product formation using arachidonic acid as substrate prein...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2018
Entry Details Article
PubMed