BDBM50206713 CHEMBL3891802

SMILES C1Cc2ccccc2N2CCCNCCC12

InChI Key InChIKey=HVGLAIHDNYRABY-UHFFFAOYSA-N

Data  3 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50206713   

Target5-hydroxytryptamine receptor 2C(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50206713(CHEMBL3891802)
Affinity DataEC50:  130nMAssay Description:Agonist activity at unedited 5-HT2C receptor (unknown origin) expressed in HEK293 cells assessed as [3H]inositol phosphate accumulation after 2 hrs b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50206713(CHEMBL3891802)
Affinity DataEC50:  126nMAssay Description:Displacement of [125I]DOI from recombinant human 5-HT2C receptor expressed in HEK293 cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2018
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50206713(CHEMBL3891802)
Affinity DataEC50:  1.00E+3nMAssay Description:Displacement of [125I]DOI from recombinant human 5-HT2B receptor expressed in HEK293 cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2018
Entry Details Article
PubMed