BDBM50207000 5-(4-bromo-5-phenylthien-3-yl)-1,2,5-thiadiazolidin-3-one 1,1-dioxide::CHEMBL241250

SMILES OC1=CN(c2csc(c2Br)-c2ccccc2)S(=O)(=O)N1

InChI Key InChIKey=NJZSZBBDUIUOMZ-UHFFFAOYSA-N

Data  1 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50207000   

TargetTyrosine-protein phosphatase non-receptor type 1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50207000(5-(4-bromo-5-phenylthien-3-yl)-1,2,5-thiadiazolidi...)
Affinity DataIC50: 2.90E+4nMAssay Description:Inhibition of PTP1B assessed as pNPP hydrolysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50207000(5-(4-bromo-5-phenylthien-3-yl)-1,2,5-thiadiazolidi...)
Affinity DataKi:  1.80E+4nMAssay Description:Inhibition of PTP1B assessed as pNPP hydrolysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed