BDBM50208729 CHEMBL3883764

SMILES N#Cc1cc2cnccc2c2[nH]c3ccccc3c12

InChI Key InChIKey=DCPBIOSSTDLFHO-UHFFFAOYSA-N

Data  2 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50208729   

TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Cnrs

Curated by ChEMBL

LigandBDBM50208729(CHEMBL3883764)Copy SMILESCopy InChI

Affinity DataIC50: 50nMAssay Description:Inhibition of GST-tagged human recombinant DYRK1A expressed in Escherichia coli using RS peptide as substrate incubated for 30 mins in presence of [g...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
9/2/2018
Entry Details Article
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TargetCyclin-dependent kinase 5 activator 1(Human)
Cnrs

Curated by ChEMBL

LigandBDBM50208729(CHEMBL3883764)Copy SMILESCopy InChI

Affinity DataIC50: 800nMAssay Description:Inhibition of human recombinant CDK5/p25 using histone H1 as substrate after 30 mins in presence of [gamma-33 P] ATP by liquid scintillation counting...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProtUniProtKB/TrEMBL
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
9/2/2018
Entry Details Article
Copy BDB DOIPubMed
Copy reaction URL