BDBM50211660 CHEMBL3915254

SMILES Cc1nc2ccccc2n(CC(=O)Nc2ccc(cc2)S(=O)(=O)NC(=S)NC2CCCCC2)c1=O

InChI Key InChIKey=WSTZIATXULQCTI-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50211660   

TargetPeroxisome proliferator-activated receptor gamma(Human)
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50211660(CHEMBL3915254)
Affinity DataIC50: 350nMAssay Description:Displacement of fluormone-PPARgamma Green from recombinant human N-terminal GST-tagged PPARgamma-LBD by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2018
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Al-Azhar University

Curated by ChEMBL
LigandPNGBDBM50211660(CHEMBL3915254)
Affinity DataIC50: 4.00E+3nMAssay Description:Displacement of fluormone-PPARgamma green from GST-tagged PPARgamma-LBD (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/15/2020
Entry Details Article
PubMed