BDBM50213309 2-(6-((5-(4-chlorophenyl)isoxazol-3-yl)methoxy)-4-methylbenzo[b]thiophen-3-yl)acetic acid::CHEMBL391085

SMILES Cc1cc(OCc2cc(on2)-c2ccc(Cl)cc2)cc2scc(CC(O)=O)c12

InChI Key InChIKey=GTZMHMRAOJUYKJ-UHFFFAOYSA-N

Data  6 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 7 hits for monomerid = 50213309   

LigandPNGBDBM50213309(2-(6-((5-(4-chlorophenyl)isoxazol-3-yl)methoxy)-4-...)
Affinity DataIC50: 311nMAssay Description:Displacement of [3H]2-(4-(2-(3-(2,4-difluorophenyl)-1-heptylureido)ethyl)phenoxy)-2-methylbutanoic acid from human PPARalpha after 30 mins by SPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50213309(2-(6-((5-(4-chlorophenyl)isoxazol-3-yl)methoxy)-4-...)
Affinity DataEC50:  638nMAssay Description:Agonist activity at human PPARdelta in HepG2 cells by GAL4-luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50213309(2-(6-((5-(4-chlorophenyl)isoxazol-3-yl)methoxy)-4-...)
Affinity DataIC50: 8.66E+3nMAssay Description:Displacement of [3H]5-(4-(3-(5-methyl-2-phenyloxazol-4-yl)propanoyl)benzyl)thiazolidine-2,4-dione from human PPARgamma after 2 hrs by SPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50213309(2-(6-((5-(4-chlorophenyl)isoxazol-3-yl)methoxy)-4-...)
Affinity DataIC50: 23nMAssay Description:Displacement of [3H]2-(4-(3-(4-acetyl-3-hydroxy-2 propyl-phenoxy)propoxy)phenoxy)acetic acid from human PPARdelta after 30 mins by SPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50213309(2-(6-((5-(4-chlorophenyl)isoxazol-3-yl)methoxy)-4-...)
Affinity DataIC50: 311nMAssay Description:Agonist activity at PPARalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
LigandPNGBDBM50213309(2-(6-((5-(4-chlorophenyl)isoxazol-3-yl)methoxy)-4-...)
Affinity DataIC50: 23.0nMAssay Description:Agonist activity at PPARdeltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
LigandPNGBDBM50213309(2-(6-((5-(4-chlorophenyl)isoxazol-3-yl)methoxy)-4-...)
Affinity DataIC50: 8.67E+3nMAssay Description:Agonist activity at PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed