BDBM50226327 CHEMBL283076

SMILES COc1c(Cl)nc(nc1NC1CCCC1)N1CCN(C)CC1

InChI Key InChIKey=ILJZSVIOWUNDKO-UHFFFAOYSA-N

Data  4 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50226327   

LigandPNGBDBM50226327(CHEMBL283076)
Affinity DataKi:  29nMAssay Description:Inhibition of [3H]idazoxan binding to alpha-2 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2018
Entry Details Article
PubMed
LigandPNGBDBM50226327(CHEMBL283076)
Affinity DataKi:  50nMAssay Description:In vitro binding affinity was measured as the inhibition of [3H]clonidine binding to alpha-2 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2018
Entry Details Article
PubMed
LigandPNGBDBM50226327(CHEMBL283076)
Affinity DataKi:  670nMAssay Description:In vitro binding affinity to Dopamine receptors of rat striatal membranes by [3H]spiroperidol displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2018
Entry Details Article
PubMed
LigandPNGBDBM50226327(CHEMBL283076)
Affinity DataKi:  1.70E+3nMAssay Description:In vitro binding affinity was measured as the inhibition of [3H]WB-4101 binding to alpha-1 adrenergic receptor of rat cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2018
Entry Details Article
PubMed