BDBM50232483 CHEMBL4061630

SMILES Cc1cc(OCc2ccccc2SC(F)(F)F)ccc1CCC(O)=O

InChI Key InChIKey=YGUAMWNBQGXDCP-UHFFFAOYSA-N

Data  4 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50232483   

TargetFree fatty acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50232483(CHEMBL4061630)
Affinity DataEC50:  1.54E+3nMAssay Description:Agonist activity at human FFA1 receptor expressed in human U2OS cells co-expressing Galpha16 assessed as calcium mobilization by Fluo-4 dye based FLI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50232483(CHEMBL4061630)
Affinity DataEC50:  1.59E+3nMAssay Description:Agonist activity at human FFA1 receptor expressed in human U2OS cells co-expressing Galpha16 assessed as calcium mobilization by Fluo-4 dye based FLI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50232483(CHEMBL4061630)
Affinity DataEC50:  794nMAssay Description:Agonist activity at human FFA4 receptor expressed in human U2OS cells co-expressing Galpha16 assessed as calcium mobilization by Fluo-4 dye based FLI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50232483(CHEMBL4061630)
Affinity DataEC50:  722nMAssay Description:Agonist activity at human FFA4 receptor expressed in human U2OS cells co-expressing Galpha16 assessed as calcium mobilization by Fluo-4 dye based FLI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details Article
PubMed