BDBM50232530 CHEMBL4098969

SMILES Cc1c(C)c(OCc2ccccc2SC(F)(F)F)ccc1CCC(O)=O

InChI Key InChIKey=TYBJCZMZWFQYBX-UHFFFAOYSA-N

Data  4 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50232530   

TargetFree fatty acid receptor 4(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50232530(CHEMBL4098969)
Affinity DataEC50:  304nMAssay Description:Agonist activity at human FFA4 receptor expressed in human U2OS cells co-expressing Galpha16 assessed as calcium mobilization by Fluo-4 dye based FLI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50232530(CHEMBL4098969)
Affinity DataEC50:  316nMAssay Description:Agonist activity at human FFA4 receptor expressed in human U2OS cells co-expressing Galpha16 assessed as calcium mobilization by Fluo-4 dye based FLI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50232530(CHEMBL4098969)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at human FFA1 receptor expressed in human U2OS cells co-expressing Galpha16 assessed as calcium mobilization by Fluo-4 dye based FLI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50232530(CHEMBL4098969)
Affinity DataEC50: <3.16E+4nMAssay Description:Agonist activity at human FFA1 receptor expressed in human U2OS cells co-expressing Galpha16 assessed as calcium mobilization by Fluo-4 dye based FLI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details Article
PubMed