BDBM50234552 CHEMBL4083160

SMILES CS(=O)(=O)NC(=O)c1cc(Cl)c(cc1F)-n1cc(F)c2cc(cnc12)-c1cccc(Cl)c1F

InChI Key InChIKey=LVGGXPAEQLLHIW-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50234552   

TargetSodium channel protein type 9 subunit alpha(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50234552(CHEMBL4083160)
Affinity DataIC50: 40nMAssay Description:Inhibition of human Nav1.7 expressed in HEK293 cells assessed as inhibition of peak current after 50 secs by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2019
Entry Details Article
PubMed