BDBM50238938 CHEMBL4095241

SMILES CC(C)(C)c1cccc(c1)-c1ccc(Oc2cccc(COc3ccccc3CCC(=O)OCCCOP(O)(=O)OC[C@H](N)C(O)=O)c2)cc1

InChI Key InChIKey=IEHHDCJODKNINL-UHFFFAOYSA-N

Data  4 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50238938   

TargetProbable G-protein coupled receptor 34(Mouse)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50238938(CHEMBL4095241)
Affinity DataEC50:  14nMAssay Description:Agonist activity at mouse GPR34 expressed in HEK293 cells co-transfected with AP-TGFalpha/chimeric Galphaq/i1 assessed as induction of ectodomain she...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 34(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50238938(CHEMBL4095241)
Affinity DataEC50:  15nMAssay Description:Agonist activity at human GPR34 expressed in HEK293 cells co-transfected with AP-TGFalpha/chimeric Galphaq/i1 assessed as induction of AP-TGFalpha re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 34(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50238938(CHEMBL4095241)
Affinity DataEC50:  15nMAssay Description:Agonist activity at human GPR34 expressed in HEK293 cells co-transfected with AP-TGFalpha/chimeric Galphaq/i1 assessed as induction of AP-TGFalpha re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 34(Mouse)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50238938(CHEMBL4095241)
Affinity DataEC50:  14nMAssay Description:Agonist activity at mouse GPR34 expressed in HEK293 cells co-transfected with AP-TGFalpha/chimeric Galphaq/i1 assessed as induction of ectodomain she...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed