BDBM50247134 1-(2-Methyl-4-(2,3,4,5-tetrahydro-1-benzazepin-1-ylcarbonyl)benzylcarbamoyl)-L-proline tertbutylester::CHEMBL462595

SMILES Cc1cc(ccc1CNC(=O)N1CCC[C@H]1C(=O)OC(C)(C)C)C(=O)N1CCCCc2ccccc12

InChI Key InChIKey=HCTXLNBEEGORFZ-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50247134   

TargetVasopressin V2 receptor(Human)
Vantia

Curated by ChEMBL
LigandPNGBDBM50247134(1-(2-Methyl-4-(2,3,4,5-tetrahydro-1-benzazepin-1-y...)
Affinity DataEC50:  390nMAssay Description:Agonist activity at human vasopressin V2 receptor expressed in HEK293 cells assessed as increase in intracellular cAMP level by CRE-luciferase report...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed