BDBM50251227 CHEMBL4084231

SMILES Cc1ccc(Oc2ccc3N(CNS(=O)(=O)c3c2)C2CC2)cc1

InChI Key InChIKey=RTQAQHMHISYJFY-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50251227   

TargetGlutamate receptor 2(Human)
University of Li£Ge

Curated by ChEMBL
LigandPNGBDBM50251227(CHEMBL4084231)
Affinity DataEC50:  3.19E+3nMAssay Description:Positive allosteric modulation of GluA2 (Q) flop isoform (unknown origin) expressed in HEK293 cells assessed as potentiation of glutamate-evoked calc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2019
Entry Details Article
PubMed
TargetGlutamate receptor 2(Human)
University of Li£Ge

Curated by ChEMBL
LigandPNGBDBM50251227(CHEMBL4084231)
Affinity DataEC50:  3.19E+3nMAssay Description:Positive allosteric modulation of GluA2 (Q) flop isoform (unknown origin) expressed in HEK293 cells assessed as potentiation of glutamate-evoked calc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2019
Entry Details Article
PubMed