BDBM50251328 CHEMBL457275::[R-(-)-Apomorphine-2-yl]-(2'-hydroxy-ethyl)ether

SMILES CN1CCc2cc(OCCO)cc-3c2[C@H]1Cc1ccc(O)c(O)c-31

InChI Key InChIKey=MLSWBRKIYGJEGT-UHFFFAOYSA-N

Data  2 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50251328   

TargetD(2) dopamine receptor(Rat)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM50251328([R-(-)-Apomorphine-2-yl]-(2'-hydroxy-ethyl)ether |...)
Affinity DataEC50:  315nMAssay Description:Agonist activity at rat dopamine D2(short) receptor expressed in CHOK1 cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM50251328([R-(-)-Apomorphine-2-yl]-(2'-hydroxy-ethyl)ether |...)
Affinity DataKi:  347nMAssay Description:Displacement of [3H]raclopride from rat dopamine D2(short) receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Mouse)
University of Debrecen

Curated by ChEMBL
LigandPNGBDBM50251328([R-(-)-Apomorphine-2-yl]-(2'-hydroxy-ethyl)ether |...)
Affinity DataKi:  5.30E+3nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in mouse Ltk- fibroblast cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed