BDBM50254163 2-(4-chlorophenylsulfonyl)-2-methyl-N-(5-o-tolyl-1,3,4-thiadiazol-2-yl)propanamide::CHEMBL461223

SMILES Cc1ccccc1-c1nnc(NC(=O)C(C)(C)S(=O)(=O)c2ccc(Cl)cc2)s1

InChI Key InChIKey=XTRAKSRSUMWOJX-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50254163   

TargetCannabinoid receptor 2(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50254163(2-(4-chlorophenylsulfonyl)-2-methyl-N-(5-o-tolyl-1...)
Affinity DataEC50:  189nMAssay Description:Agonist activity at human CB2 receptor expressed in SF9 cells assessed as inhibition of CP-55940-stimulated GTP bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50254163(2-(4-chlorophenylsulfonyl)-2-methyl-N-(5-o-tolyl-1...)
Affinity DataEC50:  1.65E+3nMAssay Description:Agonist activity at human CB1 receptor expressed in SF9 cells assessed as inhibition of CP-55940-stimulated GTP bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed