BDBM50254808 (S)-(7-(2,3-dichlorophenyl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidin-6-yl)(4-(4-fluorophenyl)piperazin-1-yl)methanone::CHEMBL480020

SMILES CC1=Nc2ccnn2[C@@H](C1C(=O)N1CCN(CC1)c1ccc(F)cc1)c1cccc(Cl)c1Cl

InChI Key InChIKey=QRLRMKZSZQUVPI-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50254808   

TargetPotassium voltage-gated channel subfamily A member 5(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50254808((S)-(7-(2,3-dichlorophenyl)-5-methyl-4,7-dihydropy...)
Affinity DataIC50: 160nMAssay Description:Inhibition of human Kv1.5 channel expressed in mouse L929 cells by EP voltage clamp techniqueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed