BDBM50256271 2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-yl)-N-(4-methoxybenzyl)acetamide::CHEMBL480539

SMILES COc1ccc(CNC(=O)Cn2nc(c(n2)-c2ccc(Cl)cc2Cl)-c2ccc(Cl)cc2Cl)cc1

InChI Key InChIKey=OPWCLDMBLALICS-UHFFFAOYSA-N

Data  2 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50256271   

TargetCannabinoid receptor 2(Human)
National Central University

Curated by ChEMBL
LigandPNGBDBM50256271(2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-...)
Affinity DataIC50: 10nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Central University

Curated by ChEMBL
LigandPNGBDBM50256271(2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-...)
Affinity DataEC50:  56.2nMAssay Description:Antagonist activity at human CB1 receptor expressed in HEK293 cells assessed as inhibition of Eu-GTP bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Central University

Curated by ChEMBL
LigandPNGBDBM50256271(2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-...)
Affinity DataIC50: 81.9nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed