BDBM50260198 CHEMBL4099403

SMILES COc1cc(Nc2ncc3CN(C(=O)N(C4CCN(CC4)C(=O)\C=C\CN(C)C)c3n2)c2c(Cl)c(OC)cc(OC)c2Cl)ccc1F

InChI Key InChIKey=CLUQPHUIWHLBAJ-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50260198   

TargetFibroblast growth factor receptor 1(Human)
Guangzhou Institutes of Biomedicine and Health

Curated by ChEMBL
LigandPNGBDBM50260198(CHEMBL4099403)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of human recombinant His-tagged FGFR1 cytoplasmic domain (308 to 731 residues) expressed in baculovirus using Tyr-4 peptide after 1 hr by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2020
Entry Details Article
PubMed