BDBM50265682 CHEMBL524089::N'-[(3Z)-6-Methoxy-1-pentyl-2-oxo-1,2-dihydro-3H-indol-3-ylidene]-2-morpholin-4-ylacetohydrazide

SMILES CCCCCN1C(=O)C(=NNC(=O)CN2CCOCC2)c2ccc(OC)cc12

InChI Key InChIKey=DJZDNOAKIJTRSE-UHFFFAOYSA-N

Data  3 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50265682   

TargetCannabinoid receptor 2(Human)
University of Montana

Curated by ChEMBL
LigandPNGBDBM50265682(N'-[(3Z)-6-Methoxy-1-pentyl-2-oxo-1,2-dihydro-3H-i...)
Affinity DataEC50:  13.3nMAssay Description:Antagonist activity at cannabinoid CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
The University of Texas M.D. Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50265682(N'-[(3Z)-6-Methoxy-1-pentyl-2-oxo-1,2-dihydro-3H-i...)
Affinity DataEC50: >1.00E+4nMAssay Description:Inverse agonist activity at human recombinant CB1 receptor expressed CHO cells membrane by [35S]GTPgamma binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Montana

Curated by ChEMBL
LigandPNGBDBM50265682(N'-[(3Z)-6-Methoxy-1-pentyl-2-oxo-1,2-dihydro-3H-i...)
Affinity DataEC50:  13.3nMAssay Description:Inverse agonist activity at human recombinant CB2 receptor expressed CHO cells membrane by [35S]GTPgamma binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed