BDBM50267947 CHEMBL4088629

SMILES Cc1cc(ccc1N)C1=NN(CC2CC(Br)=NO2)C(=O)Cc2cc3OCCOc3cc12

InChI Key InChIKey=YYXVQJJRUFHQSF-UHFFFAOYSA-N

Data  2 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50267947   

TargetGlutamate receptor 2(Human)
University of Messina

Curated by ChEMBL
LigandPNGBDBM50267947(CHEMBL4088629)
Affinity DataKi:  5.00E+4nMAssay Description:Antagonist activity at open state of GluA2Qflip isoform (unknown origin) expressed in HEK293 cells assessed as reduction in glutamate-induced current...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/1/2020
Entry Details Article
PubMed
TargetGlutamate receptor 2(Human)
University of Messina

Curated by ChEMBL
LigandPNGBDBM50267947(CHEMBL4088629)
Affinity DataKi:  5.00E+4nMAssay Description:Antagonist activity at closed state of GluA2Qflip isoform (unknown origin) expressed in HEK293 cells assessed as reduction in glutamate-induced curre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/1/2020
Entry Details Article
PubMed