BDBM50269222 CHEMBL4090974

SMILES COc1ccc(F)c(-c2ccc3c(NC(=O)c4ccc(cc4)N(C)CCN(C)C)n[nH]c3c2)c1F

InChI Key InChIKey=CGBKLNITKCQKHO-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50269222   

TargetFibroblast growth factor receptor 2(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50269222(CHEMBL4090974)
Affinity DataIC50: 35nMAssay Description:Inhibition of recombinant FGFR2 (unknown origin) using poly (Glu,Tyr)4:1 as substrate after 60 mins by ELISA based spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/9/2020
Entry Details Article
PubMed
TargetFibroblast growth factor receptor 1(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50269222(CHEMBL4090974)
Affinity DataIC50: 21nMAssay Description:Inhibition of recombinant FGFR1 (unknown origin) using poly (Glu,Tyr)4:1 as substrate after 60 mins by ELISA based spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/9/2020
Entry Details Article
PubMed