BDBM50271612 CHEMBL4127761

SMILES O=C1NC(=O)C(Cc2ccc(OCCn3cnc4ccccc34)cc2)S1

InChI Key InChIKey=PXKNQYRSNVTRNQ-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50271612   

TargetPeroxisome proliferator-activated receptor gamma(Human)
Suez Canal University

Curated by ChEMBL
LigandPNGBDBM50271612(CHEMBL4127761)
Affinity DataEC50:  2.32E+3nMAssay Description:Transactivation of recombinant human N-terminal GAL4-DBD fused PPARgamma LBD expressed in reporter cells measured after 24 hrs by luciferase reporter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Suez Canal University

Curated by ChEMBL
LigandPNGBDBM50271612(CHEMBL4127761)
Affinity DataEC50:  4.31E+3nMAssay Description:Transactivation of recombinant human FFAR1 expressed in CHOK1 cells co-expressing Galpha15 assessed as increase in calcium flux measured after 20 sec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2020
Entry Details Article
PubMed