BDBM50276174 CHEMBL4126316

SMILES CN1C(=O)CCc2ccc(NC(=O)c3ccc(c(CN4CCSCC4)c3)-c3ccccc3)cc12

InChI Key InChIKey=CWUHZJMJEKFKKO-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50276174   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Astellas Pharma

Curated by ChEMBL

LigandBDBM50276174(CHEMBL4126316)Copy SMILESCopy InChI

Affinity DataIC50: 29nMAssay Description:Displacement of [3H]RTX from human TRPV1 expressed in HEK293 cell membranes after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
5/22/2020
Entry Details Article
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