BDBM50276176 CHEMBL4127228

SMILES O=C(Nc1ccc2cccnc2c1)c1ccc(c(CN2CCCCC2)c1)-c1ccccc1

InChI Key InChIKey=DCGHAOQEKLEBHP-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50276176   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Astellas Pharma

Curated by ChEMBL

LigandBDBM50276176(CHEMBL4127228)Copy SMILESCopy InChI

Affinity DataIC50: 23nMAssay Description:Displacement of [3H]RTX from human TRPV1 expressed in HEK293 cell membranes after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
5/22/2020
Entry Details Article
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