BDBM50276181 CHEMBL4127571

SMILES O=C(Nc1ccc2oc(=O)[nH]c2c1)c1ccc(c(CN2CCCCC2)c1)-c1ccccc1

InChI Key InChIKey=DZYXAUIRFLHOHR-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50276181   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Astellas Pharma

Curated by ChEMBL

LigandBDBM50276181(CHEMBL4127571)Copy SMILESCopy InChI

Affinity DataIC50: 580nMAssay Description:Displacement of [3H]RTX from human TRPV1 expressed in HEK293 cell membranes after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
5/22/2020
Entry Details Article
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