BDBM50276196 CHEMBL4128965

SMILES O=C(Nc1ccc2CC(=O)Nc2c1)c1ccc(c(CN2CCCCC2)c1)-c1ccccc1

InChI Key InChIKey=TXDVOHJBYSDIJW-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50276196   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Astellas Pharma

Curated by ChEMBL

LigandBDBM50276196(CHEMBL4128965)Copy SMILESCopy InChI

Affinity DataIC50: 140nMAssay Description:Displacement of [3H]RTX from human TRPV1 expressed in HEK293 cell membranes after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
5/22/2020
Entry Details Article
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