BDBM50277369 CHEMBL4160688

SMILES COc1ccc(cc1)C(=O)N(Cc1ccncc1)Cc1cccc(OCc2cccc(OC)c2)c1

InChI Key InChIKey=UHWCIAZVEIMHSF-UHFFFAOYSA-N

Data  4 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50277369   

LigandPNGBDBM50277369(CHEMBL4160688)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human GLUT8 expressed in HEK293 cells transfected with GLUT1 shRNA assessed as inhibition of [3H]2-deoxy-D-glucose uptake prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandPNGBDBM50277369(CHEMBL4160688)
Affinity DataIC50: 2.85E+4nMAssay Description:Inhibition of human GLUT1 in human KMS11 cells over-expressing human GLUT1 assessed as as inhibition of receptor-mediated cell proliferation after 72...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandPNGBDBM50277369(CHEMBL4160688)
Affinity DataIC50: 1.10E+4nMAssay Description:Antagonist activity at human GLUT4 expressed in HEK293 cells transfected with GLUT1 shRNA assessed as inhibition of [3H]2-deoxy-D-glucose uptake prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed
LigandPNGBDBM50277369(CHEMBL4160688)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human GLUT1 expressed in HEK293 cells transfected with GLUT1 shRNA assessed as inhibition of [3H]2-deoxy-D-glucose uptake prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2020
Entry Details Article
PubMed