BDBM50280399 CHEMBL4172843
SMILES OC(=O)CC[C@H]1CN(c2cc(\C=C\c3c(Cl)cccc3C(F)(F)F)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F
InChI Key InChIKey=HNQAJIBKSKZNTO-UHFFFAOYSA-N
Data 5 EC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 50280399
Affinity DataEC50: 68nMAssay Description:Agonist activity at human His-tagged RORgamma-LBD expressed in Sf9 cells assessed as inhibition of N-terminal biotinylated co-activator SRC1 recruitm...More data for this Ligand-Target Pair
Affinity DataEC50: 229nMAssay Description:Agonist activity at human ROR-gamma LBD expressed in HEK293 cells assessed as transcriptional activity in presence of ursolic acid by Gal4-luciferase...More data for this Ligand-Target Pair
Affinity DataEC50: <500nMAssay Description:Agonist activity at Gal4-fused DBD RORgammat LBD (unknown origin) expressed in HEK293 cells assessed as coactivator recruitment incubated for overnig...More data for this Ligand-Target Pair
Affinity DataEC50: <500nMAssay Description:Agonist activity at His tagged RORgammat LBD (unknown origin) expressed in baculovirus infected sf9 cells assessed as biotinylated-LXXLL peptide coac...More data for this Ligand-Target Pair
Affinity DataEC50: 2.00E+3nMAssay Description:Agonist activity at human PXR-gamma expressed in HEK293 cells assessed as transcriptional activity in presence of ursolic acid by Gal4-luciferase rep...More data for this Ligand-Target Pair