BDBM50282760 CHEMBL4174996

SMILES COc1cc(OC)cc(\C=C\c2ccc3n(CCOc4ccc(CC(OCC(F)(F)F)C(O)=O)cc4)c(=O)sc3c2)c1

InChI Key InChIKey=FHWDYHYHAMRIIE-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50282760   

TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Lille

Curated by ChEMBL
LigandPNGBDBM50282760(CHEMBL4174996)
Affinity DataEC50:  20nMAssay Description:Transactivation of human Gal4-fused PPARgamma LBD expressed in African green monkey COS7 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2020
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Lille

Curated by ChEMBL
LigandPNGBDBM50282760(CHEMBL4174996)
Affinity DataEC50:  300nMAssay Description:Transactivation of human Gal4-fused PPARalpha LBD expressed in African green monkey COS7 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2020
Entry Details Article
PubMed