BDBM50283444 CHEMBL4173010

SMILES Clc1ccc(cc1)[C@H]1CN(CCN1C(=O)c1ccc(Br)cc1)C(=O)c1c[nH]c(=O)c2ccccc12

InChI Key InChIKey=XRKZUWMUFBHDMA-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50283444   

TargetEukaryotic initiation factor 4A-III(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50283444(CHEMBL4173010)
Affinity DataIC50: 290nMAssay Description:Inhibition of MLN51-induced full length recombinant human N-terminal His6/SUMO-tagged eIF4A3 RNA dependent ATPase activity expressed in Escherichia c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/4/2020
Entry Details Article
PubMed