BDBM50284097 2-Methyl-pyrazolo[1,5-a]pyridine-3-carboxylic acid (9-methyl-9-aza-bicyclo[3.3.1]non-3-yl)-amide::CHEMBL348809

SMILES CN1C2CCCC1CC(C2)NC(=O)c1c(C)nn2ccccc12

InChI Key

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50284097   

LigandPNGBDBM50284097(2-Methyl-pyrazolo[1,5-a]pyridine-3-carboxylic acid...)
Affinity DataIC50: 100nMAssay Description:Inhibition of 5-HT (1 ug/mL) induced depolarization in rat vagus nerve (5-hydroxytryptamine 3 receptor antagonism)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2012
Entry Details Article

LigandPNGBDBM50284097(2-Methyl-pyrazolo[1,5-a]pyridine-3-carboxylic acid...)
Affinity DataIC50: 64nMAssay Description:Inhibition of [3H]GR-65630 binding to rat cortical membrane serotonin 3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2012
Entry Details Article