BDBM50285231 3,5-Dihydroxy-4-(2-hydroxy-6-methoxycarbonyl-benzoyl)-benzoic acid (1R,2R)-2-(4-hydroxy-benzoylamino)-cyclopentyl ester::CHEMBL66923

SMILES COC(=O)c1cccc(O)c1C(=O)c1c(O)cc(cc1O)C(=O)O[C@@H]1CCC[C@H]1NC(=O)c1ccc(O)cc1

InChI Key InChIKey=JOOTZGPUMCZHLH-UHFFFAOYSA-N

Data  5 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50285231   

TargetProtein kinase C alpha type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM50285231(3,5-Dihydroxy-4-(2-hydroxy-6-methoxycarbonyl-benzo...)
Affinity DataIC50: 4.20E+3nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C epsilon type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM50285231(3,5-Dihydroxy-4-(2-hydroxy-6-methoxycarbonyl-benzo...)
Affinity DataIC50: 2.00E+4nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C beta type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM50285231(3,5-Dihydroxy-4-(2-hydroxy-6-methoxycarbonyl-benzo...)
Affinity DataIC50: 40nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C eta type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM50285231(3,5-Dihydroxy-4-(2-hydroxy-6-methoxycarbonyl-benzo...)
Affinity DataIC50: 400nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C delta type(Human)
Sphinx Pharmaceuticals

LigandPNGBDBM50285231(3,5-Dihydroxy-4-(2-hydroxy-6-methoxycarbonyl-benzo...)
Affinity DataIC50: 30nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article