BDBM50293263 2-(5-benzyl-2-hydroxyphenyl)-6-methyl-4H-chromen-4-one::CHEMBL522061

SMILES Cc1ccc2oc(cc(=O)c2c1)-c1cc(Cc2ccccc2)ccc1O

InChI Key InChIKey=UHHVZGAPCPFAGJ-UHFFFAOYSA-N

Data  4 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50293263   

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Lund University

Curated by ChEMBL
LigandPNGBDBM50293263(2-(5-benzyl-2-hydroxyphenyl)-6-methyl-4H-chromen-4...)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]flumazenil in rat GABAA alpha-1-beta-3-gamma-2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-5(Rat)
Lund University

Curated by ChEMBL
LigandPNGBDBM50293263(2-(5-benzyl-2-hydroxyphenyl)-6-methyl-4H-chromen-4...)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]flumazenil in rat GABAA alpha-5-beta-3-gamma-2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3(Rat)
Lund University

Curated by ChEMBL
LigandPNGBDBM50293263(2-(5-benzyl-2-hydroxyphenyl)-6-methyl-4H-chromen-4...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]flumazenil in rat GABAA alpha-3-beta-3-gamma-2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-2(Rat)
Lund University

Curated by ChEMBL
LigandPNGBDBM50293263(2-(5-benzyl-2-hydroxyphenyl)-6-methyl-4H-chromen-4...)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]flumazenil in rat GABAA alpha-2-beta-3-gamma-2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed