BDBM50293264 2-(5-bromo-2-hydroxyphenyl)-6-methylquinolin-4(1H)-one::CHEMBL452728

SMILES Cc1ccc2nc(cc(O)c2c1)-c1cc(Br)ccc1O

InChI Key InChIKey=NYRFXWGBTPDDKD-UHFFFAOYSA-N

Data  3 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50293264   

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Lund University

Curated by ChEMBL
LigandPNGBDBM50293264(2-(5-bromo-2-hydroxyphenyl)-6-methylquinolin-4(1H)...)
Affinity DataKi:  39nMAssay Description:Displacement of [3H]flumazenil in rat GABAA alpha-1-beta-3-gamma-2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3(Rat)
Lund University

Curated by ChEMBL
LigandPNGBDBM50293264(2-(5-bromo-2-hydroxyphenyl)-6-methylquinolin-4(1H)...)
Affinity DataKi:  99nMAssay Description:Displacement of [3H]flumazenil in rat GABAA alpha-3-beta-3-gamma-2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-2(Rat)
Lund University

Curated by ChEMBL
LigandPNGBDBM50293264(2-(5-bromo-2-hydroxyphenyl)-6-methylquinolin-4(1H)...)
Affinity DataKi:  120nMAssay Description:Displacement of [3H]flumazenil in rat GABAA alpha-2-beta-3-gamma-2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed