BDBM50293920 (R)-3,5-Dichloro-4-{6-chloro-4-[1-(methoxymethyl)propyl]-3-oxo-3,4-dihydropyrazin-2-ylamino}benzonitrile::CHEMBL560034

SMILES CC[C@H](COC)n1cc(Cl)nc(Nc2c(Cl)cc(cc2Cl)C#N)c1=O

InChI Key InChIKey=LKWIXUQJYZRBRT-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50293920   

TargetCorticotropin-releasing factor receptor 1(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50293920((R)-3,5-Dichloro-4-{6-chloro-4-[1-(methoxymethyl)p...)
Affinity DataIC50: 1.70nMAssay Description:Displacement of [125I]ovine-CRF from CRF1 receptor in rat frontal cortex by rapid filtration techniqueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed